文本内容:
English wordof Pharmacology钟京谕Collected by药物drug药理学pharmacology药物效应动力学pharmacodynamics药物作用drug action药物效应pharmacological effect兴奋excitation抑制inhibition特异性specificity选择性selectivity治疗作用therapeutic effect对因治疗etiological treatment对症治疗symptomatic treatment不良反应adverse drugreaction,ADR副反应side reaction毒性反应toxic reaction后遗效应residual reaction停药反应withdrawal reaction继发反应secondary reaction变态反应allergic reaction特异质反应idosyncratic reaction生理依赖性physiological dependence精神依赖性psychological dependence效量关系dose-effect relationship最小有效量/浓度minimal effectivedose/concentration阈剂量/浓度threshold dose/concentration最大效应maximal effect,Emax半最大效应浓度concentration for50%of maximaleffect,EC50效价强度potency intensity治疗指数therapeutic index,TI构效关系structure activityrelationship受体receptor亲和力affinity内在活性intrinsic activity完全激动药full agonist部分激动药partical agonist竞争性拮抗药competitive antagonist非竞争性拮抗药noncompetitive antagonist反向激动药inverse agonist药物代谢动力学pharmacokinetics,PK吸收absorption分布distribution代谢metabolism排泄excretion简单扩散simple diffusion首过消除first-pass elimination生物利用度bioavailability,BA/F生物等效性bioequivalence,BE表观分布容积apparent volumeof distribution,Vd半衰期half-life,tl/2稳态浓度steady stateconcentration抗菌谱antibacterial spectrum化疗指数chemotherapeutic index,CI最低抑菌浓度minimal inhibitoryconcentration,MIC最低杀菌浓度minimal bactericidalconcentration,MBC耐药性resistance首次接触效应first exposeeffect。